T234 Source: Uniprot

enzymeDNA polymerase gamma (PolG)

Full Name DNA polymerase gamma
Subcellular Location Mitochondrion Mitochondrion matrix, mitochondrion nucleoid

Compound Dose Time Species Model Method Result Positive criterion Reference
Emtricitabine Positive 194
Menadione 6.0 μM 1 hours human pFastBac Meassurement of DNA polymerase gamma activity Positive IC50 9
phylloquinone >200 μM 1 hours human pFastBac Meassurement of DNA polymerase gamma activity Negative IC50 9
menaquinones >200 μM 1 hours human pFastBac Meassurement of DNA polymerase gamma activity Negative IC50 9
Zalcitabine Positive 194
Didanosine Positive 194
Stavudine Positive 194
Lamivudine Positive 194
Tenofovir Positive 194
Zidovudine Positive 194
Carbovir Positive 194
Abacavir Positive 194
Fialuridine Positive 194