T019002 Source: Uniprot

protein subunitFo subunits (Fo subunits)

ATP synthase >>
Full Name Fo subunits
Subcellular Location Mitochondrion membrane Multi-pass membrane protein

Compound Dose Time Species Model Method Result Positive criterion Reference
N,N'-dicyclohexylcarbodiimide 1 mol inhibitor/mol F0 E. coli membrane H+-translocation Positive maximal inhibition 170
woodward's reagent k Positive 170
Mersalyl 130 μM bovine heart MF0, proton conductivity Positive 70% inhibition 170
Oligomycin 152 μg inhibitor/mg protein E. coli membrane vesicle, pH gradient formation Positive 170
Oligomycin 7.1 μg inhibitor/mg protein C. asciculate SMP-ATPase Positive IC50 170
Oligomycin 2.0-3.0 μg inhibitor/mg protein S. cerevisiae SMP-ATPase Positive IC50 170
Oligomycin 0.3 μM human NCI-60 cell lines F0F1-ATPase Positive IC50 170
Oligomycin 15 ng inhibitor/mg protein N. crassa SMP-ATPase Positive Ki 170
Oligomycin 0.21 μM bovine heart MF0F1-ATPase Positive Ki 170
Oligomycin 0.4 μg inhibitor/mg protein bovine heart SMP-ATPase Positive 95% inhibition 170
Oligomycin 0.5 μg/ml rat liver SMP-ATPase Positive 75% inhibition 170
ossamycin 46 μg of inhibitor/mg protein E. coli pH gradient formation by membrane vesicle Positive IC50 170
ossamycin 8 μM human NCI-60 cell lines F0F1-ATPase Positive IC50 170
ossamycin 1.3 μg of inhibitor/mg protein S. cerevisiae SMP-ATPase Positive IC50 170
venturicidin B Positive 170
Bedaquiline Positive 170
NCCD 0.65 nmol/mg protein bovine heart SMP-ATPase Positive IC50 170
NCCD 1 nmol NCCD/mg protein bovine heart SMP-ATPase Positive 85% inhibition 170
N,N'-dicyclohexylcarbodiimide 0.2 μg of inhibitor/mg protein S. cerevisiae SMP-ATPase Positive IC50 170
N,N'-dicyclohexylcarbodiimide 1-5 μg of inhibitor/mg protein T. pyriformis SMP-ATPase Positive IC50 170
N,N'-dicyclohexylcarbodiimide 200 μMa in less than 5 min and at ∼40 μMa in 30 min R. rubrum F1-ATPase Positive 170
N,N'-dicyclohexylcarbodiimide 1.9 μg/mg protein C. fasciculata SMP-ATPase Positive IC50 170
N,N'-dicyclohexylcarbodiimide 1 mol DCCD/mol F1 EF1-ATPase Positive 95% inhibition 170
N,N'-dicyclohexylcarbodiimide 30 μM membrane-bound EF0F1-ATPase Positive maximal 70-80% inhibition 170
N,N'-dicyclohexylcarbodiimide 5 μM C. thermoaceticum membrane-bound F0F1-ATPase Positive 47% inhibition 170
N,N'-dicyclohexylcarbodiimide 2 mol inhibitor bound/mol F1 bovine heart MF1-ATPase Positive 97% inhibition 170
N,N'-dicyclohexylcarbodiimide 1 mol inhibitor/mol F0 bovine heart SMP-ATPase Positive maximal inhibition 170
N,N'-dicyclohexylcarbodiimide 2 mol inhibitor/mol F0 bovine heart H+-translocation Positive maximal inhibition 170